4 Thiazolidinone Synthesis Essay

1. Akbarzadeh T, Tabatabai SA, Khoshnoud MJ, Shafaghi B, Shafiee A. Design and synthesis of 4H-3-(2-phenoxy) phenyl-1, 2, 4-triazole derivatives as benzodiazepine receptor agonists. Bioorg Med Chem. 2003;11:769–773.[PubMed]

2. Alerno S, Da Settimo F, Taliani S, Simorini F, La Motta C, Fornaciari G, et al. Medicinal chemistry of indolylglyoxylamide GABAA/BzR high affinity ligands: identification of novel anxiolytic/non sedative agents. Curr Top Med Chem. 2012;12:286–311.[PubMed]

3. Almasirad A, Hosseini R, Jalalizadeh H, Rahimi-Moghaddam Z, Abaeian N, Janafrooz M, et al. Synthesis and analgesic activity of 2-phenoxybenzoic acid and N-phenylanthranilic acid hydrazides. Biol Pharm Bull. 2006;29:1180–1185.[PubMed]

4. Almasirad A, Tabatabai SA, Faizi M, Kebriaeezadeh A, Mehrabi N, Dalvandi A, et al. Synthesis and anticonvulsant activity of new 2-substituted-5-[2-(2-fluorophenoxy) phenyl]-1, 3, 4-oxadiazoles and 1, 2, 4-triazoles. Bioorg Med Chem Lett. 2004;14:6057–6059.[PubMed]

5. Almasirad A, Vousooghi N, Tabatabai SA, Kebriaeezadeh A, Shafiee A. Synthesis, anticonvulsant and muscle relaxant activities of substituted 1, 3, 4-oxadiazole, 1, 3, 4-thiadiazole and 1, 2, 4-triazole. Acta Chim Slov. 2007;54:317–324.

6. Faizi M, Dabirian S, Tajali H, Ahmadi F, Rezaee E, Shahhosseini S, et al. Novel agonists of benzodiazepine receptors: design, synthesis, binding assay and pharmacological evaluation of 1, 2, 4-triazolo [1, 5-a] pyrimidinone and 3-amino-1, 2, 4-triazole derivatives. Bioorg Med Chem. 2015;23:480–487.[PubMed]

7. Faizi M, Sheikhha M, Ahangar N, Tabatabaei Ghomi H, Shafaghi B, Shafiee A, et al. Design, synthesis and pharmacological evaluation of novel 2-[2-(2-chlorophenoxy) phenyl]-1, 3, 4-oxadiazole derivatives as benzodiazepine receptor agonists. Iran J Pharm Res. 2012;11:83–90.[PMC free article][PubMed]

8. Grunwald C, Rundfeldt C, Lankau HJ, Arnold T, Höfgen N, Dost R, et al. Synthesis, pharmacology, and structure-activity relationships of novel imidazolones and pyrrolones as modulators of GABAA receptors. J Med Chem. 2006;49:1855–1866.[PubMed]

9. Guerrini G, Ciciani G, Cambi G, Bruni F, Selleri S, Besnard F, et al. Novel 3-iodo-8-ethoxypyrazolo [5, 1-c][1, 2, 4] benzotriazine 5-oxide as promising lead for design of a5-inverse agonist useful tools for therapy of mnemonic damage. Bioorg Med Chem. 2007;15:2573–2586.[PubMed]

10. Guerrini G, Costanzo A, Ciciani G, Bruni F, Selleri S, Costagli C, et al. Benzodiazepine receptor ligands. 8: Synthesis and pharmacological evaluation of new pyrazolo [5, 1-c][1, 2, 4] benzotriazine 5-oxide 3-and 8-disubstituted: High affinity ligands endowed with inverse-agonist pharmacological efficacy. Bioorg Med Chem. 2006;14:758–775.[PubMed]

11. Lipinski CA, Lombardo F, Dominy BW, Feeney PJ. Experimental and computational approaches to estimate solubility and permeability in drug discovery and development settings. J Adv Drug Delivery Rev. 2012;64:4–17.[PubMed]

12. Liu H, Wang L, Lv M, Pei R, Li P, Pei Z, et al. AlzPlatform: An Alzheimer’s disease domain-specific chemogenomics knowledgebase for polypharmacology and target identification research. J Chem Inf Model. 2014;54:1050–1060.[PMC free article][PubMed]

13. Mahdavi M, Akbarzadeh T, Sheibani V, Abbasi M, Firoozpour L, Tabatabai SA, et al. Synthesis of two novel 3-amino-5-[4-chloro-2-phenoxyphenyl]-4H-1, 2, 4-triazoles with anticonvulsant activity. Iranian J Pharm Res. 2010;9:265–269.[PMC free article][PubMed]

14. Rezaee E, Hedayati M, Hoghooghi Rad L, Kiani A, Shahhosseini S, Faizi M, et al. Design, synthesis and biological evaluation of some oxadiazole derivatives as novel amide-based inhibitors of soluble epoxide hydrolase. Lett Drug Des Discov. 2014;11:721–730.

15. Rezaee E, Hedayati M, Hoghooghi Rad L, Shahhosseini S, Faizi M, Tabatabai SA. Design, synthesis and biological evaluation of 4-benzamidobenzoic acid hydrazide derivatives as novel soluble epoxide hydrolase inhibitors. Iranian J Pharm Res. 2014;13:51–59.[PMC free article][PubMed]

16. Rudolph U, Knoflach F. Beyond classical benzodiazepines: novel therapeutic potential of GABAA receptor subtypes. Nat Rev Drug Discov. 2011;10:685–697.[PMC free article][PubMed]

17. Sałat K, Gawlik K, Witalis J, Pawlica-Gosiewska D, Filipek B, Solnica B, et al. Evaluation of antinociceptive and antioxidant properties of 3-[4-(3-trifluoromethyl-phenyl)-piperazin-1-yl]-dihydrofuran-2-one in mice. Arch Pharmacol. 2013;386:493–505.[PMC free article][PubMed]

18. Shingalapur RV, Hosamani KM, Keri RS, Hugar MH. Derivatives of benzimidazole pharmacophore: synthesis, anticonvulsant, antidiabetic and DNA cleavage studies. Eur J Med Chem. 2010;42:1753–1759.[PubMed]

19. Smith GB, Olsen RW. Functional domains of GABA A receptors. Trends Pharmacol Sci. 1995;16:162–168.[PubMed]

20. Tabatabai SA, Barghi Lashkari S, Zarrindast MR, Gholibeikian M, Shafiee A. Design, synthesis and anticonvulsant activity of 2-(2-phenoxy) phenyl-1, 3, 4-oxadiazole derivatives. Iran J Pharm Res. 2013;12:105–111.[PMC free article][PubMed]

21. Tripathi AC, Gupta SJ, Fatima GN, Sonar PK, Verma A, Saraf SK. 4-Thiazolidinones: the advances continue. Eur J Med Chem. 2014;72:52–77.[PubMed]

22. Zarghi A, Hajimahdi Z, Mohebbi S, Rashidi H, Mozaffari S, Sarraf S, et al. Design and synthesis of new 2-substituted-5-[2-(2-halobenzyloxy) phenyl]-1, 3, 4-oxadiazoles as anticonvulsant agents. Chem Pharm Bul. 2008;56:509–512.[PubMed]

23. Zarghi A, Hamedi S, Tootooni F, Amini B, Sharifi B, Faizi M, et al. Synthesis and pharmacological evaluation of new 2-substituted-5-{2-[(2-halobenzyl) thio) phenyl}-1, 3, 4-oxadiazoles as anticonvulsant agents. Sci Pharm. 2008;76:185–201.

24. Zarghi A, Tabatabai SA, Faizi M, Ahadian A, Navabi P, Zanganeh V, et al. Synthesis and anticonvulsant activity of new 2-substituted-5-(2-benzyloxyphenyl)-1, 3, 4-oxadiazoles. Bioorg Med Chem Lett. 2005;15:1863–1865.[PubMed]

MDPI and ACS Style

Turgut, Z.; Yolacan, C.; Aydogan, F.; Bagdatli, E.; Ocal, N. Synthesis of New Pyrazolothiazole Derivatives from 4-Thiazolidinones. Molecules2007, 12, 2151-2159.

AMA Style

Turgut Z, Yolacan C, Aydogan F, Bagdatli E, Ocal N. Synthesis of New Pyrazolothiazole Derivatives from 4-Thiazolidinones. Molecules. 2007; 12(9):2151-2159.

Chicago/Turabian Style

Turgut, Zuhal; Yolacan, Cigdem; Aydogan, Feray; Bagdatli, Emine; Ocal, Nuket. 2007. "Synthesis of New Pyrazolothiazole Derivatives from 4-Thiazolidinones." Molecules 12, no. 9: 2151-2159.

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